Kanabipiperidietanon

Kanabipiperidietanon
IUPAC ime
	2-(2-metoksifenil)-1-[1-([1-metilpiperidin-2-il]metil)indol-3-il]etanon
Identifikatori
CAS broj	1345970-43-5
ATC kod	none
ChemSpider	27330303
Hemijski podaci
Formula	C24H28N2O2
Molarna masa	376,490
	SMILES COc2ccccc2CC(=O)c(c4c1cccc4)cn1CC3CCCCN3C; ;
	InChI InChI=1S/C24H28N2O2/c1-25-14-8-7-10-19(25)16-26-17-21(20-11-4-5-12-22(20)26)23(27)15-18-9-3-6-13-24(18)28-2/h3-6,9,11-13,17,19H,7-8,10,14-16H2,1-2H3 ; Key:AJSBNWAHEDVQJT-UHFFFAOYSA-N ;

Kanabipiperidietanon (1-(N-metilpiperidin-2-ilmetil)-3-(2-metoksifenilacetil)indol) je sintetički kanabinoid koji je sastojak biljnih mešavina sintetičkih kanabisa koji su u prodaju u Japanu, zajedno sa JWH-122 i JWH-081. Njegov afinitet vezivanja (IC₅₀) za kanabinoidne receptore je 591 nM na CB₁ i 968 nM na CB₂. On je 2,3 i 9,4 puta slabiji od JWH-250 na tim biološkim ciljevima.^[1]

Reference

^ Uchiyama N, Kikura-Hanajiri R, Goda Y (2011). „Identification of a novel cannabimimetic phenylacetylindole, cannabipiperidiethanone, as a designer drug in a herbal product and its affinity for cannabinoid CB₁ and CB₂ receptors”. Chemical & Pharmaceutical Bulletin. 59 (9): 1203—5. PMID 21881274.

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Spoljašnje veze

[pmid21881274-1] Uchiyama N, Kikura-Hanajiri R, Goda Y (2011). „Identification of a novel cannabimimetic phenylacetylindole, cannabipiperidiethanone, as a designer drug in a herbal product and its affinity for cannabinoid CB₁ and CB₂ receptors”. Chemical & Pharmaceutical Bulletin. 59 (9): 1203—5. PMID 21881274.

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